1991: Young Investigator Award Sponsored by Chinese Chemistry Society of China.

2000: "Outstanding Yong Scholar's Award" by Qiu Shi Science and Technologies Foundation.

2005: "Scientific Excellence Award" by Eli Lilly and Company.

2012: National Outstanding Scientific and Technological Workers.

2016: "National Award for Natural Sciences (the Second Class)".

2021: "The Chinese Chemical Society Asymmetric Chemistry Award".

2022: "Prize for Scientific and Technological Progress" of Ho Leung Ho Lee Foundation.